Celastrol CAS 34157-83-0
Celastrol kuma milmo biyaha, wuxuu ku milmaa dimethyl sulfoxide iyo ethanol aan biyo lahayn. Waxaa laga soo qaatay maaddooyinka firfircoon ee ka hortagga kansarka ee ku jira dhirta sida Thunder God Vine iyo South Snake Vine ee qoyska Celastraceae. Waa daawo wax ku ool ah oo ka hortagta kansarka, oo la xaqiijiyay inay kiciso apoptosis unugyada kansarka iyadoo la joojinayo dhaqdhaqaaqa proteasome.
| Shay | Faahfaahinta |
| Barta karkarinta | 645.7±55.0 °C (Saadaasha) |
| Cufnaanta | 1.2 |
| Barta dhalaalaysa | 219-230°C |
| pKa | 4.78±0.70 (Saadaasha) |
| λmax | 424nm (MeOH) (iftiin) |
| Xaaladaha kaydinta | -20°C |
Celastrol waxaa loo isticmaalaa go'aaminta macluumaadka/aqoonsiga/tijaabooyinka dawooyinka, iwm. Saamaynta dawooyinka: Waxay leedahay sifooyin antioxidant oo xooggan, saameyn angiogenesis ka-hortagga kansarka, iyo saameyn ka-hortagga rheumatoid. Waa daawo wax ku ool ah oo ka hortagta proteasome, oo la xaqiijiyay inay kiciso apoptosis unugyada kansarka iyadoo la joojinayo dhaqdhaqaaqa proteasome.
Badanaa waxaa lagu buuxiyaa 25kg/durbaan, waxaana sidoo kale lagu samayn karaa xirmo gaar ah.
Celastrol CAS 34157-83-0
Celastrol CAS 34157-83-0












